Identification |
Name: | 3-Pyridinecarboxylicacid, 1-[2-[bis[4-(trifluoromethyl)phenyl]methoxy]ethyl]-1,2,5,6-tetrahydro-,hydrochloride (1:1) |
Synonyms: | 3-Pyridinecarboxylicacid, 1-[2-[bis[4-(trifluoromethyl)phenyl]methoxy]ethyl]-1,2,5,6-tetrahydro-,hydrochloride (9CI); CI 966 |
CAS: | 110283-66-4 |
Molecular Formula: | C23H21 F6 N O3 . Cl H |
Molecular Weight: | 509.87 |
InChI: | InChI=1/C23H21F6NO3.ClH/c24-22(25,26)18-7-3-15(4-8-18)20(16-5-9-19(10-6-16)23(27,28)29)33-13-12-30-11-1-2-17(14-30)21(31)32;/h2-10,20H,1,11-14H2,(H,31,32);1H |
Molecular Structure: |
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Properties |
Flash Point: | 264.7°C |
Boiling Point: | 514.1°Cat760mmHg |
Density: | g/cm3 |
Biological Activity: | Selective inhibitor of the GABA transporter GAT-1 (IC 50 values are 0.26 and 1.2 μ M at cloned human and rat GAT-1 respectively). Displays over 200-fold selectivity over GAT-2 and GAT-3. Centrally active upon systemic administration in vivo . Anticonvulsive and neuroprotective. |
Flash Point: | 264.7°C |
Safety Data |
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