Identification |
Name: | 4,8-Methano-8aH-bisbenzofuro[3,2-e:2',3'-g]isoquinoline-1,8a-diol,7-(cyclopropylmethyl)-5,6,7,8,9,14b-hexahydro-, (4bS,8R,8aS,14bR)- |
Synonyms: | 4,8-Methano-8aH-bisbenzofuro[3,2-e:2',3'-g]isoquinoline-1,8a-diol,7-(cyclopropylmethyl)-5,6,7,8,9,14b-hexahydro-, [8R-(4bS*,8a,8ab,14bb)]-; Naltriben |
CAS: | 111555-58-9 |
Molecular Formula: | C26H25 N O4 |
Molecular Weight: | 415.481 |
InChI: | InChI=1S/C26H25NO4/c28-18-8-7-15-11-20-26(29)12-17-16-3-1-2-4-19(16)30-22(17)24-25(26,21(15)23(18)31-24)9-10-27(20)13-14-5-6-14/h1-4,7-8,14,20,24,28-29H,5-6,9-13H2/t20-,24+,25+,26-/m1/s1 |
Molecular Structure: |
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Properties |
Density: | 1.5 g/cm3 |
Refractive index: | 1.779 |
Appearance: | off-white Solid |
Biological Activity: | Selective and potent δ -opioid receptor antagonist (K i values are 0.013, 19 and 152 nM for δ , μ and κ receptors respectively). Displays selectivity for the δ 2 subtype in vivo . |
Storage Temperature: | −20°C |
Color: | off-white |
Safety Data |
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