| Identification |
| Name: | Methanone,(2-amino-4,5-dimethyl-3-thienyl)[3-(trifluoromethyl)phenyl]- |
| Synonyms: | PD 81723 |
| CAS: | 132861-87-1 |
| Molecular Formula: | C14H12 F3 N O S |
| Molecular Weight: | 299.31 |
| InChI: | InChI=1/C14H12F3NOS/c1-7-8(2)20-13(18)11(7)12(19)9-4-3-5-10(6-9)14(15,16)17/h3-6H,18H2,1-2H3 |
| Molecular Structure: |
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| Properties |
| Flash Point: | 202.8°C |
| Boiling Point: | 411.7°C at 760 mmHg |
| Density: | 1.328g/cm3 |
| Refractive index: | 1.563 |
| Biological Activity: | Allosteric potentiator at the adenosine A 1 receptor; acts via agonist-dependent and -independent mechanisms. Enhances agonist affinity for, and increased t 1/2 of dissociation from, the receptor. Also inhibits basal and forskolin-stimulated adenylyl cyclase (AC) activity in A 1 receptors expressed in CHO cells, possibly via direct potentiation of constitutive receptor activity or by direct inhibition of AC. Active in vivo . |
| Flash Point: | 202.8°C |
| Storage Temperature: | −20°C |
| Color: | yellow |
| Safety Data |
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