| Identification | |
| Name: | 3-Pyridinecarboxylicacid,5-[[[3-(4,4-diphenyl-1-piperidinyl)propyl]amino]carbonyl]-1,4-dihydro-2,6-dimethyl-4-(4-nitrophenyl)-,methyl ester |
| Synonyms: | SNAP 5089 |
| CAS: | 157066-76-7 |
| Molecular Formula: | C36H40 N4 O5 |
| Molecular Weight: | 0 |
| Molecular Structure: |  |
| Properties | |
| Biological Activity: | Subtype-selective α 1A -adrenoceptor antagonist that displays > 600-fold selectivity over other adrenoceptors (K i values are 0.35, 220, 370, 540, 800 and 1200 nM for α 1A , α 1B , α 2C , α 1D , α 2B and α 2A subtypes respectively and 540 nM for L-type Ca 2+ channels). Inhibits noradrenalin-induced contractions in rabbit vascular and lower urinary tissues. |
| Safety Data | |
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