| Identification |
| Name: | Methanone, [6-iodo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)- |
| Synonyms: | AM 630;Iodopravadoline; |
| CAS: | 164178-33-0 |
| Molecular Formula: | C23H25IN2O3 |
| Molecular Weight: | 504.36 |
| InChI: | InChI=1/C23H25IN2O3/c1-16-22(23(27)17-3-6-19(28-2)7-4-17)20-8-5-18(24)15-21(20)26(16)10-9-25-11-13-29-14-12-25/h3-8,15H,9-14H2,1-2H3 |
| Molecular Structure: |
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| Properties |
| Flash Point: | 320.3°C |
| Boiling Point: | 605.9°Cat760mmHg |
| Density: | 1.49g/cm3 |
| Refractive index: | 1.646 |
| Water Solubility: | Soluble to 100 mM in DMSO |
| Solubility: | Soluble to 100 mM in DMSO |
| Appearance: | Off-white solid. |
| Biological Activity: | CB 2 antagonist/inverse agonist (K i = 31.2 nM) that displays 165-fold selectivity over CB 1 receptors. Behaves as a weak partial/inverse agonist at CB 1 receptors. |
| Flash Point: | 320.3°C |
| Safety Data |
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