| Identification |
| Name: | Phosphinic acid,P-methyl-P-(1,2,3,6-tetrahydro-4-pyridinyl)- |
| Synonyms: | Phosphinicacid, methyl(1,2,3,6-tetrahydro-4-pyridinyl)- (9CI); TPMPA |
| CAS: | 182485-36-5 |
| Molecular Formula: | C6H12 N O2 P |
| Molecular Weight: | 161.14 |
| Molecular Structure: |
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| Properties |
| Biological Activity: | A selective, competitive GABA C antagonist with only minimal effects on GABA A and GABA B receptors (K b values are 2.1 μ M (antagonist), 320 μ M (antagonist) and EC 50 ~ 500 μ M (weak agonist) respectively). Displays 8-fold selectivity for human recombinant ρ 1 receptors over ρ 2 receptors. |
| Color: | white or off-white |
| Safety Data |
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