Identification |
Name: | 1,3-BIS(4-HYDROXYPHENYL)-4-METHYL-5-[4-(2-PIPERIDINYLETHOXY)PHENOL]-1H-PYRAZOLE DIHYDROCHLORIDE |
Synonyms: | METHYL-PIPERIDINO-PYRAZOLE DIHYDROCHLORIDE;1,3-BIS(4-HYDROXYPHENYL)-4-METHYL-5-[4-(2-PIPERIDINYLETHOXY)PHENOL]-1H-PYRAZOLE DIHYDROCHLORIDE;MPP DIHYDROCHLORIDE;MMP DIHYDROCHLORIDE;MPP2HCl;Methyl-piperidino-pyrazole, 1,3-Bis(4-hydroxyphenyl)-4-methyl-5-[4-(2-piperidinylethoxy)phenol]-1H-pyrazole dihydrochloride |
CAS: | 289726-02-9 |
Molecular Formula: | C29H33Cl2N3O3 |
Molecular Weight: | 542.5 |
Molecular Structure: |
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Properties |
Biological Activity: | Selective, high affinity silent antagonist at ERa receptors. Displays > 200-fold selectivity for ERa over ERb. K i values are 2.7 and 1800 nM at ERa and ERb receptors respectively. |
Safety Data |
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