Identification |
Name: | 1-Pentanone,1-[3-(2-aminoethyl)-2-(phenylmethyl)-1H-indol-1-yl]- |
Synonyms: | 1H-Indole-3-ethanamine,1-(1-oxopentyl)-2-(phenylmethyl)- (9CI); DH 97 |
CAS: | 343263-95-6 |
Molecular Formula: | C22H26 N2 O |
Molecular Weight: | 334.45 |
Molecular Structure: |
|
Properties |
Biological Activity: | A relatively potent MT 2 melatonin receptor antagonist (pK i value = 8.03), displaying 89- and 229-fold selectivity over MT 1 and GPR50 (melatonin-related orphan receptor) respectively. |
Safety Data |
|
|