Identification |
Name: | Trisoxireno[4b,5:6,7:8a,9]phenanthro[1,2-c]furan-1(3H)-one,3b,4,4a,6,6a,7a,7b,8b,9,10-decahydro-6-hydroxy-8b-methyl-6a-(1-methylethyl)-,(3bS,4aS,5aS,6R,6aR,7aS,7bS,8aS,8bS)- |
Synonyms: | (-)-Triptolide;NSC 163062;PG 490;[3bS-(3ba,4aa,5aR*,6b,6ab,7ab,7ba,8aR*,8bb)]-3b,4,4a,6,6a,7a,7b,8b,9,10-Decahydro-6-hydroxy-8b-methyl-6a-(1-methylethyl)trisoxireno[4b,5:6,7:8a,9]phenanthro[1,2-c]furan-1(3H)-one; |
CAS: | 38748-32-2 |
Molecular Formula: | C20H24O6 |
Molecular Weight: | 360.40096 |
InChI: | InChI=1S/C20H24O6/c1-8(2)18-13(25-18)14-20(26-14)17(3)5-4-9-10(7-23-15(9)21)11(17)6-12-19(20,24-12)16(18)22/h8,11-14,16,22H,4-7H2,1-3H3/t11-,12-,13-,14-,16+,17-,18-,19+,20+/m0/s1 |
Molecular Structure: |
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Properties |
Density: | 1.48 g/cm3 |
Refractive index: | 1.647 |
Water Solubility: | DMSO: soluble |
Solubility: | DMSO: soluble |
Appearance: | white to off-white solid |
Biological Activity: | Inhibits cytokine-induced gene expression via inhibition of NF- κ B transcriptional activity. Induces apoptosis in tumor cells by blocking TNF- α mediated c-IAP2 and c-IAP1 (members of the inhibitor of apoptosis family) induction. Immunosuppressive with anti-inflammatory and antitumor activity. |
Storage Temperature: | 2-8°C |
Color: | white to off-white |
Usage: | Diterpenoid triepoxide with immunosuppressant and antitumor properties. |
Safety Data |
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