Identification |
Name: | 2-Propenamide,N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[4-(1,1-dimethylethyl)phenyl]-, (2E)- |
Synonyms: | (2E)-N-(2H,3H-Benzo[3,4-e]-1,4-dioxan-6-yl)-3-[4-(tert-butyl)phenyl]prop-2-enamide;AMG 9810; |
CAS: | 545395-94-6 |
Molecular Formula: | C21H23NO3 |
Molecular Weight: | 337.41 |
InChI: | InChI=1/C21H23NO3/c1-21(2,3)16-7-4-15(5-8-16)6-11-20(23)22-17-9-10-18-19(14-17)25-13-12-24-18/h4-11,14H,12-13H2,1-3H3,(H,22,23)/b11-6+ |
Molecular Structure: |
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Properties |
Flash Point: | 263.8°C |
Boiling Point: | 512.5°C at 760 mmHg |
Density: | 1.175g/cm3 |
Refractive index: | 1.617 |
Biological Activity: | Potent and selective, competitive vanilloid TRPV1 receptor antagonist (IC 50 = 17 nM). Inhibits capsaicin-, proton-, heat- and endogenous ligand-induced activation of human and rat recombinant TRPV1 receptors. Displays antihyperalgesic properties in a rat model of inflammatory pain. |
Flash Point: | 263.8°C |
Storage Temperature: | 2-8°C |
Safety Data |
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