Identification |
Name: | 2-[[4-(2-PYRIDINYL)-1-PIPERAZINYL]METHYL]-1H-BENZIMIDAZOLE TRIHYDROCHLORIDE |
Synonyms: | ABT 724 TRIHYDROCHLORIDE;2-[[4-(2-PYRIDINYL)-1-PIPERAZINYL]METHYL]-1H-BENZIMIDAZOLE TRIHYDROCHLORIDE |
CAS: | 70006-24-5 |
Molecular Formula: | C17H22Cl3N5 |
Molecular Weight: | 402.74908 |
InChI: | InChI=1/C17H19N5/c1-2-6-15-14(5-1)19-16(20-15)13-21-9-11-22(12-10-21)17-7-3-4-8-18-17/h1-8H,9-13H2,(H,19,20) |
Molecular Structure: |
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Properties |
Flash Point: | 285.6°C |
Boiling Point: | 548.6°C at 760 mmHg |
Density: | 1.275g/cm3 |
Refractive index: | 1.687 |
Biological Activity: | Potent dopamine D 4 receptor partial agonist (EC 50 = 12.4 nM; 61% efficacy vs. dopamine). Has no agonist activity at D 2 receptors (EC 50 > 10 μ M). Selective in rats in vivo : produces penile erection following i.c.v. administration; increases intracavernosal pressure and potentiates the proerectile effects of sildenafil following s.c. administration. Displays minimal side effects. |
Flash Point: | 285.6°C |
Safety Data |
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