Identification |
Name: | Bicyclo[3.1.0]hexane-1-methanol,4-[2-iodo-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, 1-(dihydrogenphosphate), (1R,2S,4S,5S)- |
Synonyms: | Bicyclo[3.1.0]hexane-1-methanol,4-[2-iodo-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, dihydrogenphosphate (ester), (1R,2S,4S,5S)- (9CI); MRS 2500 |
CAS: | 779323-43-2 |
Molecular Formula: | C13H18 I N5 O8 P2 |
Molecular Weight: | 0 |
Molecular Structure: |
![(C13H18IN5O8P2) Bicyclo[3.1.0]hexane-1-methanol,4-[2-iodo-6-(methylamino)-9H-purin-9-yl]-2-(phosphonooxy)-, dihydrog...](https://img1.guidechem.com/chem/e/dict/10/779323-43-2.jpg) |
Properties |
Biological Activity: | Highly potent and selective antagonist of the platelet P2Y 1 receptor (K i = 0.78 nM). Inhibits ADP-induced aggregation of human platelets with an IC 50 value of 0.95 nM. Prevents thrombus formation in vivo . |
Safety Data |
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