| Identification |
| Name: | 6-[5-[(2S)-2-AZETIDINYLMETHOXY]-3-PYRIDINYL]-5-HEXYN-1-OL DIHYDROCHLORIDE |
| Synonyms: | 6-[5-[(2S)-2-AZETIDINYLMETHOXY]-3-PYRIDINYL]-5-HEXYN-1-OL DIHYDROCHLORIDE;SAZETIDINE A DIHYDROCHLORIDE |
| CAS: | 820231-95-6 |
| Molecular Formula: | C15H22Cl2N2O2 |
| Molecular Weight: | 0 |
| Molecular Structure: |
![(C15H22Cl2N2O2) 6-[5-[(2S)-2-AZETIDINYLMETHOXY]-3-PYRIDINYL]-5-HEXYN-1-OL DIHYDROCHLORIDE;SAZETIDINE A DIHYDROCHLORI...](https://img.guidechem.com/structure/820231-95-6.gif) |
| Properties |
| Biological Activity: | Subtype-selective α 4 β 2 nicotinic acetylcholine receptor ligand (K i values are 0.26 and 54 nM at α 4 β 2 and α 3 β 4 receptors respectively). May act as a silent desensitizer or as an agonist (EC 50 = 1.1 nM for nAChR-stimulated dopamine release). Exhibits analgesic activity in vivo . |
| Safety Data |
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