| Identification |
| Name: | 5,6-DIHYDRO-5-METHYL-6-OXO-4H-IMIDAZO[1,5-A]THIENO[2,3-F][1,4]DIAZEPINE-3-CARBOXYLIC ACID 1,1-DIMETHYLETHYL ESTER |
| Synonyms: | RO 19-4603;5,6-DIHYDRO-5-METHYL-6-OXO-4H-IMIDAZO[1,5-A]THIENO[2,3-F][1,4]DIAZEPINE-3-CARBOXYLIC ACID 1,1-DIMETHYLETHYL ESTER;5,6-Dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a]thieno[2,3-f][1,4]diazepine-3-carboxylicacid1,1-dimethylethylester |
| CAS: | 99632-94-7 |
| Molecular Formula: | C15H17N3O3S |
| Molecular Weight: | 319.38 |
| InChI: | InChI=1/C15H17N3O3S/c1-15(2,3)21-14(20)11-10-7-17(4)13(19)12-9(5-6-22-12)18(10)8-16-11/h5-6,8H,7H2,1-4H3 |
| Molecular Structure: |
![(C15H17N3O3S) RO 19-4603;5,6-DIHYDRO-5-METHYL-6-OXO-4H-IMIDAZO[1,5-A]THIENO[2,3-F][1,4]DIAZEPINE-3-CARBOXYLIC ACID...](https://img.guidechem.com/structure/99632-94-7.gif) |
| Properties |
| Flash Point: | 279°C |
| Boiling Point: | 537.7°C at 760 mmHg |
| Density: | 1.37g/cm3 |
| Refractive index: | 1.659 |
| Biological Activity: | Benzodiazepine inverse agonist. Binds with high affinity to both diazepam-sensitive (DS) and diazepam-insensitive (DI) GABA A receptors (K i values are ~ 0.2 and ~ 2.6 nM for DS and DI receptors respectively). Antagonizes effects of ethanol on locomotor behavior and suppresses ethanol intake in alcohol-preferring rats. |
| Flash Point: | 279°C |
| Safety Data |
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