Identification |
Name: | Methanesulfonamide,N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]-1-piperidinyl]ethyl]-,hydrochloride (1:1) |
Synonyms: | Methanesulfonamide,N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]-1-piperidinyl]ethyl]-,monohydrochloride (9CI); RS 67506 |
CAS: | 168986-61-6 |
Molecular Formula: | C18H28 Cl N3 O4 S . Cl H |
Molecular Weight: | 454.41 |
InChI: | InChI=1/C18H28ClN3O4S.ClH/c1-26-18-12-16(20)15(19)11-14(18)17(23)4-3-13-5-8-22(9-6-13)10-7-21-27(2,24)25;/h11-13,21H,3-10,20H2,1-2H3;1H |
Molecular Structure: |
|
Properties |
Flash Point: | 320.8°C |
Boiling Point: | 606.9°C at 760 mmHg |
Biological Activity: | A potent and selective 5-HT 4 partial agonist, with a pK i of 8.8 at 5-HT 4 sites in guinea pig striatum, but < 6.0 at several other receptors including 5-HT 1A, 1D, 2A, 2C , D 1 , D 2 and M 1-3 . It is active in vivo and has an intrinsic activity compared to 5-HT of 0.6. |
Flash Point: | 320.8°C |
Safety Data |
|
|