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Bromocriptine mesylate (22260-51-1)

Identification
Name:Bromocriptine mesylate
Synonyms:Bromocriptine mesilate (JP14);Bromocriptine mesylate (USP);Bromergon;Parlodel (TN);Pravidel;Prestwick_771;Ergotaman-3,6,18-trione, 2-bromo-12-hydroxy-2-(1-methylethyl)-5- (2-methylpropyl)-, (5alpha)-;2-Bromo-alpha-ergocryptine methanesulfonate;Bromocryptine mesylate;Parlodel;CB 154;Ergotaman-3',6',18-trione,2-bromo-12'- hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)-,(5'R)-,monomethanesulfonate (salt);Bagren;
CAS:22260-51-1
EINECS: 244-881-1
Molecular Formula: C32H40BrN5O5.CH4SO3
Molecular Weight: 654.5945
InChI: InChI=1S/C32H40BrN5O5/c1-16(2)12-24-29(40)37-11-7-10-25(37)32(42)38(24)30(41)31(43-32,17(3)4)35-28(39)18-13-20-19-8-6-9-22-26(19)21(27(33)34-22)14-23(20)36(5)15-18/h6,8-9,13,16-18,23-25,34,42H,7,10-12,14-15H2,1-5H3,(H,35,39)/t18-,23-,24+,25+,31-,32+/m1/s1
Molecular Structure: (C32H40BrN5O5.CH4SO3) Bromocriptine mesilate (JP14);Bromocriptine mesylate (USP);Bromergon;Parlodel (TN);Pravidel;Prestwic...
Properties
Water Solubility:H2O: 0.8 mg/mL
Solubility:H2O: 0.8 mg/mL
Appearance:white solid
Specification:

 Bromocriptine mesylate (CAS NO.22260-51-1) also can be called Parlodel ; 2-Bromine-a-ergocryptine Methanesulfonate ; 8,9-hexahydroindolo[4,3-fg]quinoléine-9-carboxamide (1:1) ; 2-Bromo-12'-hydroxy-5'a-isobutyl-2'-isopropylergotaman-3',6',18-trione Monomethanesulphonate .

Biological Activity: Selective D 2 -like dopamine receptor agonist (K i values are ~ 8, ~ 5, ~ 290, ~ 440 and ~ 450 nM for D 2 , D 3 , D 4 , D 1 and D 5 receptors respectively).
Storage Temperature: 2-8°C
Color: white
Usage:Dopamine receptor agonist; derivative of the ergotoxin group of ergot alkaloids. Prolactin inhibitor; antiparkinsonian.
Safety Data
Hazard Symbols Xn: Harmful