Identification |
Name: | Bromocriptine mesylate |
Synonyms: | Bromocriptine mesilate (JP14);Bromocriptine mesylate (USP);Bromergon;Parlodel (TN);Pravidel;Prestwick_771;Ergotaman-3,6,18-trione, 2-bromo-12-hydroxy-2-(1-methylethyl)-5- (2-methylpropyl)-, (5alpha)-;2-Bromo-alpha-ergocryptine methanesulfonate;Bromocryptine mesylate;Parlodel;CB 154;Ergotaman-3',6',18-trione,2-bromo-12'- hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)-,(5'R)-,monomethanesulfonate (salt);Bagren; |
CAS: | 22260-51-1 |
EINECS: | 244-881-1 |
Molecular Formula: | C32H40BrN5O5.CH4SO3 |
Molecular Weight: | 654.5945 |
InChI: | InChI=1S/C32H40BrN5O5/c1-16(2)12-24-29(40)37-11-7-10-25(37)32(42)38(24)30(41)31(43-32,17(3)4)35-28(39)18-13-20-19-8-6-9-22-26(19)21(27(33)34-22)14-23(20)36(5)15-18/h6,8-9,13,16-18,23-25,34,42H,7,10-12,14-15H2,1-5H3,(H,35,39)/t18-,23-,24+,25+,31-,32+/m1/s1 |
Molecular Structure: |
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Properties |
Water Solubility: | H2O: 0.8 mg/mL |
Solubility: | H2O: 0.8 mg/mL |
Appearance: | white solid |
Specification: |
Bromocriptine mesylate (CAS NO.22260-51-1) also can be called Parlodel ; 2-Bromine-a-ergocryptine Methanesulfonate ; 8,9-hexahydroindolo[4,3-fg]quinoléine-9-carboxamide (1:1) ; 2-Bromo-12'-hydroxy-5'a-isobutyl-2'-isopropylergotaman-3',6',18-trione Monomethanesulphonate .
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Biological Activity: | Selective D 2 -like dopamine receptor agonist (K i values are ~ 8, ~ 5, ~ 290, ~ 440 and ~ 450 nM for D 2 , D 3 , D 4 , D 1 and D 5 receptors respectively). |
Storage Temperature: | 2-8°C |
Color: | white |
Usage: | Dopamine receptor agonist; derivative of the ergotoxin group of ergot alkaloids. Prolactin inhibitor; antiparkinsonian. |
Safety Data |
Hazard Symbols |
Xn: Harmful
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