Identification |
Name: | 5H-Thiazolo[3,2-a]pyrimidin-5-one,6-[2-[4-[bis(4-fluorophenyl)methylene]-1-piperidinyl]ethyl]-7-methyl- |
Synonyms: | Ritanserin;Tiserton |
CAS: | 87051-43-2 |
Molecular Formula: | C27H25 F2 N3 O S |
Molecular Weight: | 477.58 |
InChI: | InChI=1/C27H25F2N3OS/c1-18-24(26(33)32-16-17-34-27(32)30-18)12-15-31-13-10-21(11-14-31)25(19-2-6-22(28)7-3-19)20-4-8-23(29)9-5-20/h2-9,16-17H,10-15H2,1H3 |
Molecular Structure: |
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Properties |
Flash Point: | 328°C |
Boiling Point: | 618.7°C at 760 mmHg |
Density: | 1.3g/cm3 |
Refractive index: | 1.646 |
Specification: | usageEng:A potent 5-HT2A serotonin receptor antagonist/inverse agonist that crosses the blood-brain barrier. Safety Statements:22-26-36 22:Do not breathe dust 26:In case of contact with eyes, rinse immediately with plenty
of water and seek medical advice 36:Wear suitable protective clothing |
Biological Activity: | Potent and long-acting 5-HT 2 receptor antagonist (K i = 0.39 nM). Anxiolytic in vivo . |
Flash Point: | 328°C |
Color: | white |
Usage: | A potent 5-HT2A serotonin receptor antagonist/inverse agonist that crosses the blood-brain barrier. |
Safety Data |
Hazard Symbols |
Xi: Irritant
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