Identification |
Name: | 5,8,11,14-Eicosatetraenamide,N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-, (5Z,8Z,11Z,14Z)- |
Synonyms: | 5,8,11,14-Eicosatetraenamide,N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-, (all-Z)-; N-Arachidonoylserotonin |
CAS: | 187947-37-1 |
Molecular Formula: | C30H42 N2 O2 |
Molecular Weight: | 462.67 |
Molecular Structure: |
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Properties |
Biological Activity: | Dual fatty acid amide hydrolase (FAAH) inhibitor/TRPV1 antagonist (IC 50 values are 5.6 μ M and 37-40 nM for FAAH and TRPV1 respectively). Inactive at cPLA 2 , CB 1 or 5-HT receptors. Displays strong analgesic activity against both acute and chronic peripheral pain. |
Storage Temperature: | −20°C |
Safety Data |
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